CN104892668B - 考布他汀类似物水溶性前‑前药及其制备方法 - Google Patents
考布他汀类似物水溶性前‑前药及其制备方法 Download PDFInfo
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CN108607605A (zh) * | 2018-06-11 | 2018-10-02 | 徐州得铸生物科技有限公司 | 一种用于合成异戊烯酸甲酯的催化剂 |
CN112898128B (zh) * | 2021-02-08 | 2023-07-07 | 苏州华道生物药业股份有限公司 | 红褐林蚁信息素成分3-乙基-4-甲基戊醇的合成方法 |
Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
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US5561122A (en) * | 1994-12-22 | 1996-10-01 | Arizona Board Of Regents Acting On Behalf Of Arizona State University | Combretastatin A-4 prodrug |
WO2002006279A1 (en) * | 2000-07-17 | 2002-01-24 | Oxigene Inc | Efficient method of synthesizing combretastatin a-4 prodrugs |
CN101220054A (zh) * | 2008-01-29 | 2008-07-16 | 成都恒基医药科技有限公司 | 康普瑞汀a-4磷酸酯二钠盐的制备方法 |
CN102015620A (zh) * | 2008-02-28 | 2011-04-13 | 赛诺菲-安万特 | 制备考布他汀的方法 |
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EP1299337A4 (en) * | 2000-04-27 | 2004-10-13 | Univ Arizona State | HYDROXYPHENSTATIN AND ITS PROMEDICATIONS |
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Patent Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
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US5561122A (en) * | 1994-12-22 | 1996-10-01 | Arizona Board Of Regents Acting On Behalf Of Arizona State University | Combretastatin A-4 prodrug |
WO2002006279A1 (en) * | 2000-07-17 | 2002-01-24 | Oxigene Inc | Efficient method of synthesizing combretastatin a-4 prodrugs |
CN101220054A (zh) * | 2008-01-29 | 2008-07-16 | 成都恒基医药科技有限公司 | 康普瑞汀a-4磷酸酯二钠盐的制备方法 |
CN102015620A (zh) * | 2008-02-28 | 2011-04-13 | 赛诺菲-安万特 | 制备考布他汀的方法 |
Non-Patent Citations (2)
Title |
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R.Brown et al..Carbon-14 radiosynthesis of combretastatinA-1 (CA1) and its corresponding phosphate prodrug (CA1P).《J. Label Compd. Radiopharm》.2009,第52卷(第14期),第567-570页. * |
夏虎雄等.考布他汀4A 磷酸酯缓释纳米粒的制备及抗肿瘤活性考察.《中国实验方剂学杂志》.2013,第19卷(第8期),第40-43页. * |
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